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HRH3

HRH3,即組胺受體H3,別名組胺H3受體。它是一種G蛋白偶聯(lián)受體(GPCR)家族成員,主要在中樞神經(jīng)系統(tǒng)的組胺能神經(jīng)元上表達,同時也在免疫細胞等外周組織中發(fā)揮作用。HRH3的作用機制主要涉及調(diào)節(jié)神經(jīng)遞質(zhì)的合成和釋放,它在突觸前作為自身受體抑制組胺的合成和分泌,在突觸后作為異源受體調(diào)節(jié)其他神經(jīng)遞質(zhì)的活性。HRH3的激活可以影響多種生理過程,包括睡眠-覺醒周期、食欲、認知功能以及腦缺血等。HRH3在生物學(xué)上的意義非常廣泛,它不僅參與調(diào)節(jié)中樞神經(jīng)系統(tǒng)的功能,還與多種疾病的發(fā)生發(fā)展相關(guān)。例如,在肝臟中,HRH3的表達水平與肝細胞癌的發(fā)展有關(guān)。此外,HRH3還涉及到自身免疫性疾病,如多發(fā)性硬化癥,其在神經(jīng)源性控制中整合了外周炎癥信號。HRH3的功能異常與精神分裂癥等精神疾病的陰性癥狀和認知功能有關(guān),因此,HRH3拮抗劑的開發(fā)為這些疾病的治療提供了新的策略。

熱銷產(chǎn)品

HRH3 Recombinant Monoclonal Antibody (CSB-RA783626A0HU)

驗證數(shù)據(jù)

CSB-RA783626A0HU

Overlay Peak curve showing SH-SY5Y cells surface stained with CSB-RA783626A0HU (red line) at 1:50. Then 10% normal goat serum to block non-specific protein-protein interactions followed by the antibody (1μg/1*106cells) for 45min at 4℃. The secondary antibody used was FITC-conjugated Goat Anti-rabbit IgG(H+L) at 1:200 dilution for 35min at 4℃.Control antibody (green line) was rabbit IgG (1μg/1*106cells) used under the same conditions. Acquisition of >10,000 events was performed.

HRH3 Antibody (CSB-PA897568LA01HU)

驗證數(shù)據(jù)

CSB-PA897568LA01HU

Western Blot
Positive WB detected in: A549 whole cell lysate
All lanes: HRH3 antibody at 2.5µg/ml
Secondary
Goat polyclonal to rabbit IgG at 1/50000 dilution
Predicted band size: 49, 50, 41, 48, 37, 46 kDa
Observed band size: 49 kDa

CSB-PA897568LA01HU

Immunohistochemistry of paraffin-embedded human brain tissue using CSB-PA897568LA01HU at dilution of 1:100

CSB-PA897568LA01HU

Immunofluorescent analysis of A549 cells using CSB-PA897568LA01HU at dilution of 1:100 and Alexa Fluor 488-congugated AffiniPure Goat Anti-Rabbit IgG(H+L)

HRH3 Antibodies

HRH3 for Homo sapiens (Human)

HRH3 Proteins

HRH3 Proteins for Mus musculus (Mouse)

HRH3 Proteins for Cavia porcellus (Guinea pig)

HRH3 Proteins for Rattus norvegicus (Rat)

HRH3 Proteins for Homo sapiens (Human)



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