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FOLR1

FOLR1(葉酸受體1)是一種成人葉酸受體,也稱為葉酸結合蛋白(FBP),由FOLR1基因編碼。這種膜結合糖蛋白對葉酸和幾種還原葉酸衍生物具有高親和力,主要功能是介導5-甲基四氫葉酸的細胞內運輸,對細胞生長和增殖至關重要。FOLR1的結構包括跨膜結構域,并存在膜結合和可溶性兩種形式。 除了在葉酸轉運中的基本作用外,FOLR1還參與了多種信號通路,包括JAK-STAT3、ERK1/2信號通路,并可能作為轉錄因子參與基因表達調控。FOLR1在Wnt和ERK信號通路中發揮作用,通過增加活性β-catenin、磷酸化ERK以及Wnt和ERK調控基因的表達。此外,FOLR1還可能參與Wnt和TGFβ信號通路。 FOLR1的異常表達與多種癌癥的發生、發展密切相關,其在腫瘤細胞中的高表達通常與癌癥進展加快和患者預后不良有關。因此,FOLR1不僅是癌癥治療研究中的潛在靶點,而且在葉酸受體靶向治療領域具有重要的應用前景。


熱銷產品

Recombinant Human Folate receptor alpha(FOLR1),partial (Active) (CSB-MP008784HU1)

驗證數據

CSB-MP008784HU1

(Tris-Glycine gel) Discontinuous SDS-PAGE (reduced) with 5% enrichment gel and 15% separation gel.

CSB-MP008784HU1

Activity
Measured by its binding ability in a functional ELISA. Immobilized human FOLR1 at 2 μg/ml can bind Anti-FOLR1 recombinant antibody(CSB-RA008784MA1HU). The EC50 is 6.893-7.883 ng/mL.

CSB-MP008784HU1

The purity of FOLR1 was greater than 95% as determined by SEC-HPLC

Recombinant Macaca fascicularis Folate receptor alpha(FOLR1),partial (Active) (CSB-MP5002MOV)

驗證數據

CSB-MP5002MOV

(Tris-Glycine gel) Discontinuous SDS-PAGE (reduced) with 5% enrichment gel and 15% separation gel.

CSB-MP5002MOV

Activity
Measured by its binding ability in a functional ELISA. Immobilized Cynomolgus FOLR1 at 2 μg/ml can bind Anti-FOLR1 recombinant antibody(CSB-RA008784MA1HU). The EC50 is 2.900-3.544 ng/mL.

FOLR1 Antibodies

FOLR1 for Homo sapiens (Human)

FOLR1 Proteins

FOLR1 Proteins for Homo sapiens (Human)

FOLR1 Proteins for Mus musculus (Mouse)

FOLR1 Proteins for Bos taurus (Bovine)

FOLR1 ELISA Kit

FOLR1 ELISA Kit for Homo sapiens (Human)