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SLC7A5

SLC7A5全稱為溶質(zhì)載體家族7成員5(Solute Carrier Family 7 Member 5),也被稱為L(zhǎng)型氨基酸轉(zhuǎn)運(yùn)蛋白1(LAT1)或CD98輕鏈。SLC7A5主要通過(guò)與SLC3A2(CD98重鏈)結(jié)合形成異源二聚體,負(fù)責(zé)轉(zhuǎn)運(yùn)細(xì)胞必需的中性氨基酸如亮氨酸、苯丙氨酸等,其活性與細(xì)胞增殖、代謝調(diào)控密切相關(guān)。LAT1在多種惡性腫瘤中異常高表達(dá),通過(guò)激活mTORC1信號(hào)網(wǎng)絡(luò)促進(jìn)腫瘤生長(zhǎng)、侵襲及化療耐藥,尤其在膠質(zhì)瘤、乳腺癌和結(jié)直腸癌中成為預(yù)后不良的標(biāo)志物。近年來(lái)針對(duì)LAT1的小分子抑制劑開(kāi)發(fā)進(jìn)展顯著,例如JPH203已在肝癌和胰腺癌模型中顯示抗腫瘤效果,KYT-0353等候選藥物也進(jìn)入臨床前研究階段。SLC7A5與血腦屏障的氨基酸運(yùn)輸功能關(guān)聯(lián),其異常表達(dá)還可能參與神經(jīng)系統(tǒng)疾病如癲癇的病理過(guò)程。

熱銷產(chǎn)品

Recombinant Human Large neutral amino acids transporter small subunit 1 (SLC7A5), partial (CSB-EP021717HU)

驗(yàn)證數(shù)據(jù)

CSB-EP021717HU

(Tris-Glycine gel) Discontinuous SDS-PAGE (reduced) with 5% enrichment gel and 15% separation gel.

SLC7A5 Antibody (CSB-PA068714)

驗(yàn)證數(shù)據(jù)

CSB-PA068714

Gel: 6%SDS-PAGE,Lysate: 40 μg,,Primary antibody: CSB-PA068714(SLC7A5 Antibody) at dilution 1/300 dilution,Secondary antibody: Goat anti rabbit IgG at 1/8000 dilution,Exposure time: 10 seconds

SLC7A5 Antibodies

SLC7A5 for Homo sapiens (Human)

SLC7A5 Proteins

SLC7A5 Proteins for Homo sapiens (Human)

SLC7A5 Proteins for Rattus norvegicus (Rat)

SLC7A5 Proteins for Oryctolagus cuniculus (Rabbit)

SLC7A5 Proteins for Homo sapiens (Human)