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MYC

MYC全稱為myelocytomatosis oncogene,又名c-Myc、v-myc或BHLHE39,是調控細胞增殖的核心轉錄因子。MYC通過結合MAX蛋白形成異源二聚體,特異性識別DNA的E-box序列,激活涉及細胞周期進程、代謝重編程和凋亡抑制的靶基因表達。其在胚胎發育和組織再生中起關鍵作用,異常激活可導致超過70%的人類腫瘤發生,包括伯基特淋巴瘤、神經母細胞瘤和多種實體瘤。Wnt、Notch等發育通路常與MYC形成調控網絡,而PI3K/AKT/mTOR通路則介導其促癌效應。
當前針對MYC的直接抑制劑尚未上市,但通過表觀遺傳調控的BET蛋白抑制劑(如OTX015)已進入血液腫瘤的II期臨床試驗。小分子化合物MYCi975通過破壞MYC/MAX相互作用進入臨床前研究,同時針對MYC蛋白穩定性的aurora激酶抑制劑Alisertib在乳腺癌治療中顯示出協同效應。反義寡核苷酸藥物如AZD9150曾嘗試阻斷MYC mRNA,但因療效有限終止研發。近年來CRISPR基因編輯技術和PROTAC降解劑為靶向MYC提供了新思路,其中MTX-216等候選藥物正在評估中。

熱銷產品

Recombinant Human Myc proto-oncogene protein (MYC),Biotinylated (CSB-EP015270HU-B)

驗證數據

CSB-EP015270HU-B

(Tris-Glycine gel) Discontinuous SDS-PAGE (reduced) with 5% enrichment gel and 15% separation gel.

MYC Recombinant Monoclonal Antibody (CSB-RA914333A0HU)

驗證數據

CSB-RA914333A0HU

Overlay histogram showing Hela cells stained with CSB-RA914333A0HU (red line) at 1:50. The cells were fixed with 70% Ethylalcohol (18h) and then incubated in 10% normal goat serum to block non-specific protein-protein interactions followedby the antibody (1μg/1*106 cells) for 1 h at 4℃.The secondary antibody used was FITC-conjugated goat anti-rabbit IgG (H+L) at 1/200 dilution for 30min at 4℃. Control antibody (green line) was Rabbit IgG (1μg/1*106 cells) used under the same conditions. Acquisition of >10,000 events was performed.

Human c-myc Oncogene product,c-myc ELISA Kit (CSB-E09260h)

驗證數據

CSB-E09260h 標準曲線

貨號:CSB-E09260h

規格:96T/48T

靈敏度:0.078 ng/mL

檢測范圍:0.312 ng/mL-20 ng/mL

These standard curves are provided for demonstration only. A standard curve should be generated for each set of samples assayed.

MYC Antibodies

MYC for Mus musculus (Mouse)

MYC for Homo sapiens (Human)

MYC Proteins

MYC Proteins for Felis catus (Cat) (Felis silvestris catus)

MYC Proteins for Mus musculus (Mouse)

MYC Proteins for Gallus gallus (Chicken)

MYC Proteins for Homo sapiens (Human)

MYC Proteins for Rattus norvegicus (Rat)

MYC Proteins for Macaca mulatta (Rhesus macaque)

MYC Proteins for Marmota monax (Woodchuck)

MYC Proteins for Pan troglodytes (Chimpanzee)

MYC Proteins for Callithrix jacchus (White-tufted-ear marmoset)

MYC Proteins for Hylobates lar (Common gibbon)

MYC Proteins for Pan paniscus (Pygmy chimpanzee) (Bonobo)

MYC Proteins for Pongo pygmaeus (Bornean orangutan)

MYC Proteins for Feline leukemia virus

MYC Proteins for Avian retrovirus MH2

MYC Proteins for Avian myelocytomatosis virus CMII

MYC Proteins for Avian retrovirus OK10

MYC Proteins for Feline leukemia virus FTT

MYC Proteins for Carassius auratus (Goldfish)

MYC Proteins for Avian myelocytomatosis virus HBI

MYC Proteins for Oncorhynchus mykiss (Rainbow trout) (Salmo gairdneri)

MYC Proteins for Avian myelocytomatosis virus MC29

MYC Proteins for Avian retrovirus MH2E21

MYC Proteins for Asterias rubens (Common European starfish) (Asterias vulgaris)

MYC Proteins for Canis familiaris (Dog) (Canis lupus familiaris)

MYC Proteins for Ovis aries (Sheep)

MYC Proteins for Sus scrofa (Pig)

MYC Proteins for Bos taurus (Bovine)

MYC Proteins for Sylvilagus floridanus (Cottontail rabbit)

MYC Proteins for Pteropus hypomelanus (Island flying fox) (Variable flying fox)

MYC Proteins for Galeopterus variegatus (Malayan flying lemur) (Cynocephalus variegatus)

MYC Proteins for Tupaia glis (Tree shrew)

MYC Proteins for Tadarida brasiliensis (Brazilian free-tailed bat)

MYC Proteins for Drosophila melanogaster (Fruit fly)

MYC ELISA Kit

MYC ELISA Kit for Homo sapiens (Human)



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