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ANTXR1

ANTXR1全稱為炭疽毒素受體1(Anthrax Toxin Receptor 1),早期研究中被稱為腫瘤內(nèi)皮標記物8(TEM8)。ANTXR1屬于Ⅰ型跨膜蛋白家族,通過特異性結(jié)合炭疽桿菌毒素的保護性抗原組分,介導毒素進入宿主細胞,成為炭疽感染的關(guān)鍵分子靶點。近年來研究發(fā)現(xiàn),TEM8在正常生理狀態(tài)下參與血管新生調(diào)控,其胞外段含有的血管性血友病因子A結(jié)構(gòu)域(VWA)可與膠原蛋白等細胞外基質(zhì)成分相互作用,影響內(nèi)皮細胞遷移和血管網(wǎng)絡(luò)形成。
在疾病領(lǐng)域,ANTXR1的異常表達與多種實體瘤密切相關(guān),例如結(jié)直腸癌、乳腺癌中常出現(xiàn)蛋白高表達,可能通過促進腫瘤血管生成加速癌癥進展。臨床前研究表明,針對TEM8的單克隆抗體或小分子抑制劑可顯著抑制小鼠模型中腫瘤生長和轉(zhuǎn)移。此外,ANTXR1突變與罕見的GAPO綜合征相關(guān),表現(xiàn)為生長遲緩、脫發(fā)及骨發(fā)育異常。目前基于該靶點的藥物研發(fā)主要集中在炭疽毒素中和劑和抗腫瘤生物制劑兩大方向,已有數(shù)款單抗藥物進入Ⅰ/Ⅱ期臨床試驗階段。

熱銷產(chǎn)品

Recombinant Human Anthrax toxin receptor 1 (ANTXR1), partial (CSB-YP001832HU)

驗證數(shù)據(jù)

CSB-YP001832HU

(Tris-Glycine gel) Discontinuous SDS-PAGE (reduced) with 5% enrichment gel and 15% separation gel.

ANTXR1 Antibody (CSB-PA001832ESR1HU)

驗證數(shù)據(jù)

CSB-PA001832ESR1HU

Immunohistochemistry of paraffin-embedded human lung cancer using CSB-PA001832ESR1HU at dilution of 1:100

Human anthrax toxin receptor 1(ANTXR1) ELISA kit (CSB-EL001832HU)

驗證數(shù)據(jù)

CSB-EL001832HU 標準曲線

貨號:CSB-EL001832HU

規(guī)格:96T/48T

靈敏度:15.6 pg/mL

檢測范圍:62.5 pg/mL-4000 pg/mL

These standard curves are provided for demonstration only. A standard curve should be generated for each set of samples assayed.

ANTXR1 Antibodies

ANTXR1 for Homo sapiens (Human)

ANTXR1 Proteins

ANTXR1 Proteins for Homo sapiens (Human)

ANTXR1 Proteins for Mus musculus (Mouse)

ANTXR1 Proteins for Rattus norvegicus (Rat)

ANTXR1 ELISA Kit

ANTXR1 ELISA Kit for Homo sapiens (Human)