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ADAMTS4

ADAMTS4蛋白全稱為整合素樣金屬蛋白酶與血小板反應蛋白基序4,常被稱為Aggrecanase-1或ADMP-1。該蛋白在維持細胞外基質動態平衡中起關鍵作用,能夠特異性分解軟骨組織中的核心成分aggrecan,這種特性使其成為關節退行性疾病的重要研究靶點。在骨關節炎和類風濕性關節炎患者體內,其異常活躍的酶切活性會加速軟骨基質破壞,導致關節結構塌陷和功能喪失。ADAMTS4在腫瘤微環境中同樣扮演著特殊角色,可能通過重塑細胞外基質促進癌細胞侵襲轉移,特別是在乳腺癌和膠質瘤中觀察到其表達水平與疾病進展密切相關。
針對ADAMTS4的藥物開發主要聚焦于選擇性抑制劑研究,已有多個小分子化合物進入臨床前試驗階段,通過阻斷其酶活性來減緩軟骨退化進程。其中部分黃酮類衍生物在動物模型中顯示出保護關節軟骨的效果,而基于單克隆抗體的靶向療法也取得突破性進展。值得關注的是,某些已上市的抗炎藥物被發現具有間接調控該蛋白活性的潛能,這為老藥新用開辟了新方向。目前相關研究正在探索其在神經退行性疾病中的應用價值,特別是阿爾茨海默病中淀粉樣斑塊的形成可能與ADAMTS4介導的蛋白水解過程存在關聯。

熱銷產品

Recombinant Human A disintegrin and metalloproteinase with thrombospondin motifs 4 (ADAMTS4), partial (CSB-EP001311HU1)

驗證數據

CSB-EP001311HU1

(Tris-Glycine gel) Discontinuous SDS-PAGE (reduced) with 5% enrichment gel and 15% separation gel.

ADAMTS4 Antibody (CSB-PA001311LA01HU)

驗證數據

CSB-PA001311LA01HU

Immunohistochemistry of paraffin-embedded human heart tissue using CSB-PA001311LA01HU at dilution of 1:100

CSB-PA001311LA01HU

Western Blot
Positive WB detected in: Mouse kidney tissue
All lanes: ADAMTS4 antibody at 3.2µg/ml
Secondary
Goat polyclonal to rabbit IgG at 1/50000 dilution
Predicted band size: 91 kDa
Observed band size: 91 kDa

CSB-PA001311LA01HU

Immunohistochemistry of paraffin-embedded human liver tissue using CSB-PA001311LA01HU at dilution of 1:100

CSB-PA001311LA01HU

IHC image of CSB-PA001311LA01HU diluted at 1:250 and staining in paraffin-embedded human lung tissue performed on a Leica BondTM system. After dewaxing and hydration, antigen retrieval was mediated by high pressure in a citrate buffer (pH 6.0). Section was blocked with 10% normal goat serum 30min at RT. Then primary antibody (1% BSA) was incubated at 4°C overnight. The primary is detected by a biotinylated secondary antibody and visualized using an HRP conjugated SP system.

Human ADAM metallopeptidase with thrombospondin type 1 motif4,ADAMTS4 ELISA Kit (CSB-E11848h)

驗證數據

CSB-E11848h 標準曲線

貨號:CSB-E11848h

規格:96T/48T

靈敏度:3.125 ng/ml

檢測范圍:12.5 ng/ml - 800 ng/ml

These standard curves are provided for demonstration only. A standard curve should be generated for each set of samples assayed.

ADAMTS4 Antibodies

ADAMTS4 for Homo sapiens (Human)

ADAMTS4 Proteins

ADAMTS4 Proteins for Homo sapiens (Human)

ADAMTS4 ELISA Kit

ADAMTS4 ELISA Kit for Homo sapiens (Human)



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